> Trialight public data. Index of pages: https://trialight.com/llms.txt
> Web page: https://trialight.com/data/asset/lb-102-4fafa13e-2b6e-4289-b389-c2f1e2b594e9
> Record changed: 2026-10-13

# LB-102

Highest phase reached

Phase 2

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

Drug type

Small molecule

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

## Development status

**Listing at source**

Listed

**Highest phase reached**

Phase 2

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

## Names and chemistry

**Drug type**

Small molecule

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

**Drug name**

LB-102

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

**Molecular weight**

383.51

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

**Structure (SMILES)**

CCN1CCCC1CNC(=O)c1cc(S(=O)(=O)CC)c(NC)cc1OC

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

### Other names (11)

- lb 102
- Lb-102
- LB-102
- LB-102 (100 mg tablet)
- LB-102 (50 mg tablet)
- lb102
- LB102
- n methyl amisulpride
- n methylamisulpride
- N'-methyl amisulpride
- N'-methylamisulpride

## Identifiers

**CAS registry numbers**

- 2227154-23-4

**ChEMBL ID**

CHEMBL4594422

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

**InChIKey**

NXKXZXNNWRYXRE-UHFFFAOYSA-N

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL4594422)

**PubChem compound IDs**

- 134542980

**FDA ingredient codes (UNII)**

- N81WKW91XF

## Regulatory information

### Other regulatory facts

**First in class**

No

**Orphan designation**

No

## Pharmacology

### Investigated indications

- **Condition**  
Schizophrenia

**Highest recorded phase**  
2

**Condition identifier**  
MONDO:0005090

**Subject identifier**  
D012559

### Open Targets indications (4)

- **Condition identifier**  
EFO\_0007634

**Highest recorded phase**  
2
- **Condition identifier**  
EFO\_0009963

**Highest recorded phase**  
2
- **Condition identifier**  
MONDO\_0005090

**Highest recorded phase**  
2
- **Condition identifier**  
MONDO\_0005090

**Highest recorded phase**  
3

### Trial references (3)

- NCT04187560  
Source: [clinicaltrials.gov](https://clinicaltrials.gov/study/NCT04187560)
- NCT04588129  
Source: [clinicaltrials.gov](https://clinicaltrials.gov/study/NCT04588129)
- NCT06179108  
Source: [clinicaltrials.gov](https://clinicaltrials.gov/study/NCT06179108)

## Chemical properties

**Hydrogen bond acceptors**

6

**Hydrogen bond donors**

2

**Polar surface area**

87.74

**Calculated partition coefficient (ALogP)**

1.74

**Calculated partition coefficient (XLogP)**

2.1

**Prodrug**

No

**Chirality**

Racemic

**Inorganic**

No

**Rule-of-five violations**

0

**Rotatable bonds**

8

**Heavy atoms**

26

**Molecular formula**

C18H29N3O4S

**Monoisotopic mass**

383.18787759

**Natural product**

No

## Evidence counts

**Recorded assays**

4

**Active assays**

4

### Active assay types

- Confirmatory

## Related records

### Trials (448)

- 52-week Open Label Safety-Tolerability Study
- A Bioavailability Study Comparing 3 Different AZD1981 Tablets
- A Clinical Evaluation on Traditional Chinese Medicine Diagnosis and Treatment Program Blocking and Reversing Hepatitis B-related Liver Fibrosis - a Randomized, Controlled, Double-blind, Multi-center Clinical Trial
- A Clinical Intervention Study of Tangningtongluo on Diabetic Foot Ulcer
- A Clinical Study Comparing the Bioavailability of HRS-2189 Tablets
- A Clinical Study of HRS-5765 in Healthy Participants
- A Clinical Study of HRS-8364 in the Treatment of Advanced Solid Tumor Subjects
- A Clinical Study on the Safety and Efficacy of GP681 Tablets in the Treatment of Uncomplicated Acute Influenza
- A Clinical Study to Assess the Safety and Effectiveness of Herbal Supplement in Adult Human Subjects.
- A Clinical Study to Evaluate the Efficacy and Safety of D-2570 in the Treatment of Moderate to Severe Plaque Psoriasis
- A Clinical Study to Evaluate the Efficacy and Safety of HRS9531 Tablets in Overweight or Obese Subjects
- [A Clinical Study to Evaluate the Long-term Safety of HRS-1893 in Hypertrophic Cardiomyopathy](https://trialight.com/data/trial/a-clinical-study-to-evaluate-the-long-term-safety-of-hrs-9f6191c7-54bf-40c6-9199-501244b86f1e.md)
- A Clinical Study to Explore Biomarkers for Drug-induced Liver Injury (DILI)
- A Clinical Trial for Azvudine in the Treatment of Novel Coronavirus Pneumonia (COVID-19）
- A Clinical Trial of HRS-3095 in Patients With Chronic Spontaneous Urticaria
- A Clinical Trial of TQB3455 Tablets in Patients With Hematological Malignancies
- A Clinical Trial of XZP-6019 Tablets in Healthy Subjects
- A Clinical Trial on the Safety and Efficacy of TQB3909 Tablets in Patients With Recurrent or Refractory Chronic Lymphocytic Leukemia (CLL) /Small Lymphocytic Lymphoma (SLL) .
- A Clinical Trial to Assess Three Different Doses of OPS-2071 in Patients With Bacterial Enteritis
- A Comparative Pharmacokinetic Study of Single-Dose Administration of HR091506 Tablets From Different Batches in Healthy Subjects

### In development for (1)

- [Schizophrenia](https://trialight.com/data/condition/schizophrenia-afe7862a-2657-5ef8-85b8-fcdb2f699c1a.md) Phase 2

---

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