> Trialight public data. Index of pages: https://trialight.com/llms.txt
> Web page: https://trialight.com/data/asset/azilsartan-mepixetil-fd55358a-3aa9-4021-ab98-638ad5716aee
> Record changed: 2026-11-04

# Azilsartan mepixetil

Highest phase reached

Phase 2

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

Drug type

Small molecule

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

## Development status

**Listing at source**

Listed

**Highest phase reached**

Phase 2

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

## Names and chemistry

**Drug type**

Small molecule

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

**Drug name**

Azilsartan mepixetil

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

**Molecular weight**

678.7

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

**Structure (SMILES)**

CCOc1nc2cccc(C(=O)OC(C)OC(=O)OCc3nc(C)c(C)nc3C)c2n1Cc1ccc(-c2ccccc2-c2nc(=O)o\[nH\]2)cc1

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

### Other names (6)

- azilsartan mepixetil
- Azilsartan mepixetil
- azilsartan mepixetil \[INN\]
- azilsartan mepixetil inn
- qr 01019
- QR-01019

## Identifiers

**CAS registry numbers**

- 1596357-16-2

**ChEMBL ID**

CHEMBL5095053

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

**InChIKey**

JXSDNNVNQNYJSP-UHFFFAOYSA-N

Source: [www.ebi.ac.uk](https://www.ebi.ac.uk/chembl/explore/compound/CHEMBL5095053)

**PubChem compound IDs**

- 137091385

**FDA ingredient codes (UNII)**

- C2GK4G74Y7

## Regulatory information

### Other regulatory facts

**First in class**

No

**Orphan designation**

No

## Pharmacology

### Drug classification

**Drug name stem**

\-sartan

## Chemical properties

**Hydrogen bond acceptors**

13

**Hydrogen bond donors**

1

**Polar surface area**

173.55

**Calculated partition coefficient (ALogP)**

6.07

**Calculated partition coefficient (XLogP)**

6.1

**Prodrug**

No

**Chirality**

Racemic

**Inorganic**

No

**Rule-of-five violations**

3

**Rotatable bonds**

11

**Heavy atoms**

50

**Molecular formula**

C36H34N6O8

**Monoisotopic mass**

678.24381206

**Natural product**

No

## Related records

### Trials (1)

- [A Phase II Clinical Study of QR12000 Compound Tablets in Patients With Moderate to Severe Essential Hypertension](https://trialight.com/data/trial/a-phase-ii-clinical-study-of-qr12000-compound-tablets-in-039e8548-5a65-4507-be36-db003c696d2e.md)

---

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